SCHEMBL7700574

SCHEMBL7700574

O=C(O)Nc1cc(COC2CCCCO2)c(-c2ccccc2F)cc1[N+](=O)[O-]

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.38
RAB9A P51151 4/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
NPC1 O15118 3/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
HCAR3 P49019 2/20 0.38
MAPT P10636 5/20 0.36
CREBBP Q92793 2/20 0.36
EP300 Q09472 1/20 0.36
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 4/20 0.34
MEN1 O00255 2/20 0.34
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7139514 0.90 CHRM3 (0.35) ALDH1A1RAB9ASMN1; SMN2NPC1L3MBTL1
SCHEMBL7703580 0.87 HCAR3 (0.38) ALDH1A1RAB9ASMN1; SMN2NPC1L3MBTL1
SCHEMBL7700560 0.86 CREBBP (0.37) ALDH1A1RAB9ASMN1; SMN2NPC1CREBBP
SCHEMBL7698563 0.82 HCAR3 (0.40) ALDH1A1RAB9ASMN1; SMN2NPC1L3MBTL1
SCHEMBL7139585 0.77 MMP8 (0.35) ALDH1A1L3MBTL1HCAR3MAPTCREBBP
SCHEMBL7704396 0.76 CREBBP (0.34) CREBBPEP300KMT2AMEN1
SCHEMBL7141267 0.76 HDAC3 (0.37) ALDH1A1RAB9ASMN1; SMN2NPC1CREBBP
SCHEMBL7147995 0.73 ALDH1A1 (0.36) ALDH1A1RAB9ASMN1; SMN2NPC1L3MBTL1
SCHEMBL5563454 0.73 KMT2A (0.38) ALDH1A1SMN1; SMN2L3MBTL1HCAR3MAPT
SCHEMBL7140551 0.71 HCAR3 (0.36) ALDH1A1RAB9ASMN1; SMN2NPC1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224174-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001029011-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-26 WO disclosed