SCHEMBL7699016

SCHEMBL7699016

CSc1nccn1-c1cccc(C(=O)CC(=O)Nc2cc(-c3ccccc3F)c(OC(C)(C)C)cc2NC(=O)O)c1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TP53 P04637 5/20 0.41
MAPT P10636 2/20 0.40
TSHR P16473 2/20 0.38
LMNA P02545 4/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7143546 0.93 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2TP53MAPTTSHR
SCHEMBL7704777 0.91 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2TP53MAPTTSHR
SCHEMBL7146199 0.85 ALDH1A1 (0.38) ALDH1A1SMN1; SMN2TP53MAPTTSHR
SCHEMBL7704182 0.84 CYP3A4 (0.35) ALDH1A1SMN1; SMN2TP53MAPTTSHR
SCHEMBL7705335 0.83 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2TP53MAPTTSHR
SCHEMBL7703856 0.81 CYP3A4 (0.37) ALDH1A1SMN1; SMN2TP53MAPTTSHR
SCHEMBL7141959 0.79 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2TP53MAPTTSHR
SCHEMBL7703510 0.78 VCP (0.41)
SCHEMBL7704530 0.78 DHODH (0.37) ALDH1A1
SCHEMBL7704536 0.77 DHODH (0.36) ALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224174-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001029011-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-26 WO disclosed