SCHEMBL7704536

SCHEMBL7704536

CC(C)(C)Oc1cc(NC(=O)O)c(NC(=O)CC(=O)c2ccnc(C#N)c2)cc1-c1ccccc1F

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 4/20 0.36
PARP14 Q460N5 1/20 0.34
RAB9A P51151 3/20 0.34
ALDH1A1 P00352 2/20 0.34
NPC1 O15118 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KMT2A Q03164 5/20 0.33
MEN1 O00255 3/20 0.33
MAPT P10636 2/20 0.32
CTSA P10619 1/20 0.32
CHEK1 O14757 1/20 0.32
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7141050 0.92 CYP17A1 (0.35) DHODHPARP14RAB9AALDH1A1NPC1
SCHEMBL7704530 0.86 DHODH (0.37) DHODHRAB9AALDH1A1KMT2AMEN1
SCHEMBL7140010 0.85 MEN1 (0.36) DHODHPARP14ALDH1A1KMT2AMEN1
SCHEMBL7703510 0.80 VCP (0.41)
SCHEMBL7145193 0.80 CYP17A1 (0.37)
SCHEMBL7704777 0.79 ALDH1A1 (0.39) RAB9AALDH1A1NPC1SMN1; SMN2MAPT
SCHEMBL7702829 0.79 GAA (0.37) DHODHRAB9ANPC1SMN1; SMN2KMT2A
SCHEMBL5868818 0.79 CYP17A1 (0.41) PARP14MAPT
SCHEMBL7704182 0.78 CYP3A4 (0.35) RAB9AALDH1A1SMN1; SMN2KMT2AMEN1
SCHEMBL7145960 0.78 EGLN2 (0.36) DHODHALDH1A1KMT2AMEN1PDCD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224174-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001029011-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-26 WO disclosed