SCHEMBL770091

SCHEMBL770091

CCCCNC(=O)CCCC(=O)N1CCCC2CCCCC21

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
PRCP P42785 2/20 0.42
DPP4 P27487 3/20 0.40
ACE P12821 3/20 0.39
ACE2 Q9BYF1 3/20 0.39
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL770870 0.97 OPRD1 (0.47) OPRD1NPSR1PRCPDPP4ACE
SCHEMBL769971 0.96 OPRD1 (0.46) OPRD1NPSR1PRCPDPP4
SCHEMBL770182 0.94 OPRD1 (0.49) OPRD1PRCPDPP4
SCHEMBL770458 0.94 OPRD1 (0.40) OPRD1NPSR1PRCPDPP4
SCHEMBL770224 0.91 OPRD1 (0.43) OPRD1PRCPDPP4
SCHEMBL770644 0.88 EPHX1 (0.44) NPSR1
SCHEMBL770987 0.86 NPSR1 (0.44) NPSR1DPP4GAA
SCHEMBL770672 0.86 DRD2 (0.40) OPRD1NPSR1PRCPDPP4
SCHEMBL17690765 0.85 MEN1 (0.49)
SCHEMBL771646 0.82 ALDH1A1 (0.51) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2439202-B1 INHIBITOR COMPOUNDS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 SALVAT LAB SA (ES) 2016-04-20 EP disclosed
US-8822452-B2 Inhibitor compounds of 11-beta-hydroxysteroid dehydrogenase type 1 LABORATORIOS SALVAT, S.A. (ES) 2014-09-02 US disclosed
US-20130303522-A1 INHIBITOR COMPOUNDS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 LABORATORIOS SALVAT, S.A. (ES) 2013-11-14 US disclosed
US-8524894-B2 Inhibitor compounds of 11-beta-hydroxysteroid dehydrogenase type 1 LABORATORIOS SALVAT, S.A. (ES) 2013-09-03 US disclosed
US-20120071466-A1 INHIBITOR COMPOUNDS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 LABORATORIOS SALVAT, S.A. (ES) 2012-03-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130303522-A1 INHIBITOR COMPOUNDS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 HSD11B1, HSD17B1, HSD11B2 OPRD1 942/4885NPSR1 1890/4885PRCP 1922/4885
US-20120071466-A1 INHIBITOR COMPOUNDS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 HSD11B1, HSD17B1, HSD11B2 OPRD1 945/4885NPSR1 1896/4885PRCP 1940/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.