SCHEMBL7701231

SCHEMBL7701231

N#Cc1c(Br)n(CCc2ccc(F)cc2)c2ncnc(N)c12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.55
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 2/20 0.47
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
LRRK2 Q5S007 10/20 0.45
ADORA2A P29274 2/20 0.42
ADORA1 P30542 1/20 0.42
NSD2 O96028 1/20 0.37
NSD3 Q9BZ95 1/20 0.37
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RET P07949 1/20 0.35
CDK5 Q00535 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7699518 0.88 KDM4E (0.57) DYRK1AKDM4EALDH1A1GLAGAA
SCHEMBL7697867 0.88 DYRK1A (0.54) DYRK1AKDM4EALDH1A1GLAGAA
SCHEMBL7696582 0.88 DYRK1A (0.57) DYRK1AKDM4ELRRK2ADORA2AADORA1
SCHEMBL7701233 0.87 DYRK1A (0.51) DYRK1AKDM4EALDH1A1GLAGAA
SCHEMBL7700915 0.84 DYRK1A (0.50) DYRK1ALRRK2ADORA2AADORA1
SCHEMBL7701581 0.82 DYRK1A (0.55) DYRK1AKDM4ELRRK2ADORA2AADORA1
SCHEMBL7700326 0.79 LRRK2 (0.52) DYRK1AKDM4EALDH1A1GLAGAA
SCHEMBL7695781 0.79 DYRK1A (0.56) DYRK1AKDM4ELRRK2ADORA2AADORA1
SCHEMBL7699589 0.78 DYRK1A (0.55) DYRK1AKDM4ELRRK2ADORA2AADORA1
SCHEMBL7702669 0.77 DYRK1A (0.57) DYRK1AKDM4EGAALRRK2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6342501-B1 VIRICIDES THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2002-01-29 US disclosed