SCHEMBL7701458

SCHEMBL7701458

CC(C)(C)OC(=O)N1C(=O)C(Cc2ccc(-c3ccc(F)cc3)cc2)C[C@H]1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 1/20 0.38
KLK7 P49862 6/20 0.38
HDAC1 Q13547 2/20 0.37
HDAC2 Q92769 2/20 0.37
ROCK2 O75116 1/20 0.37
P2RX7 Q99572 2/20 0.36
KLK5 Q9Y337 5/20 0.36
HTT P42858 1/20 0.35
BACE1 P56817 1/20 0.35
BACE2 Q9Y5Z0 1/20 0.35
GPR119 Q8TDV5 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PRSS1 P07477 2/20 0.35
PRSS2 P07478 2/20 0.35
PRSS3 P35030 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7699900 0.91 KLK7 (0.43) KLK7KLK5GPR119KMT2APRSS1
SCHEMBL31486428 0.87 KLK7 (0.49) KLK7P2RX7KLK5MEN1KMT2A
SCHEMBL8669568 0.87 KLK7 (0.49) KLK7P2RX7KLK5MEN1KMT2A
SCHEMBL5065670 0.87 KLK7 (0.49) KLK7P2RX7KLK5MEN1KMT2A
SCHEMBL1371651 0.84 PPARG (0.41) KLK7P2RX7KLK5
SCHEMBL1371650 0.84 PPARG (0.41) KLK7P2RX7KLK5
SCHEMBL2185219 0.83 PPARG (0.45) P2RX7HTTMEN1KMT2A
SCHEMBL8211740 0.82 ROCK2 (0.38) MMP13ROCK2P2RX7HTT
SCHEMBL5204187 0.82 OPRK1 (0.44) KLK7P2RX7KLK5
SCHEMBL27840720 0.80 P2RX7 (0.41) P2RX7HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002014261-A2 4-SUBSTITUTED D-GLUTAMIC ACID DERIVATIVES FOR USE AS ANTIBIOTIC ELI LILLY AND COMPANY (US) 2002-02-21 WO disclosed