SCHEMBL7701561

SCHEMBL7701561

O=C(C=Cc1ccccc1Cl)N1CCC(CN2CCC(c3c[nH]c4ccc(O)cc34)CC2)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 16/20 0.61
SLC2A1 P11166 1/20 0.55
HTR1A P08908 1/20 0.49
DRD2 P14416 1/20 0.49
HTR1B P28222 1/20 0.49
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
HTR1E P28566 1/20 0.49
HTR1F P30939 1/20 0.49
HTR7 P34969 1/20 0.49
DRD3 P35462 1/20 0.49
HTR2B P41595 1/20 0.49
HTR6 P50406 1/20 0.49
CCR5 P51681 1/20 0.49
MAPT P10636 1/20 0.49
BLM P54132 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703004 0.87 CCR2 (0.76) CCR2SLC2A1HTR1ADRD2HTR1B
SCHEMBL7701558 0.81 CCR2 (0.57) CCR2SLC2A1HTR1ADRD2HTR1B
SCHEMBL7702549 0.80 SLC2A1 (0.82) CCR2SLC2A1
SCHEMBL7703003 0.77 CCR2 (0.62) CCR2SLC2A1HTR1ADRD2HTR1B
SCHEMBL2902532 0.72 L3MBTL1 (0.67) CCR2MAPT
SCHEMBL7701609 0.71 CCR2 (0.75) CCR2SLC2A1HTR1ADRD2HTR1B
SCHEMBL7700302 0.71 SLC2A1 (0.66) CCR2SLC2A1
SCHEMBL7532398 0.71 OPRM1 (0.77) DRD2HTR1BMAPTBLMNPSR1
SCHEMBL7694623 0.71 CCR2 (0.68) CCR2SLC2A1HTR1ADRD2HTR1B
SCHEMBL7694620 0.70 CCR2 (0.56) CCR2SLC2A1HTR1ADRD2HTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002079190-A1 3-SUBSTITUTED INDOLES AS CHEMOKINE ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-10-10 WO disclosed