SCHEMBL7701596

SCHEMBL7701596

NC(=O)Nc1ccc2[nH]cc(C3CCN(CC4CCN(/C=C/C(=O)c5ccc(Cl)c(Cl)c5)CC4)CC3)c2c1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 7/20 0.51
HTR1D P28221 13/20 0.49
HTR1B P28222 10/20 0.49
CHRM2 P08172 1/20 0.47
DRD2 P14416 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7699076 0.93 CCR2 (0.52) CCR2HTR1DHTR1BCHRM2DRD2
SCHEMBL7695961 0.92 HTR1D (0.54) CCR2HTR1DHTR1BCHRM2DRD2
SCHEMBL7695531 0.89 CCR2 (0.52) CCR2HTR1DHTR1BDRD2
SCHEMBL7703003 0.88 CCR2 (0.62) CCR2HTR1DHTR1BDRD2
SCHEMBL7696192 0.88 CCR2 (0.58) CCR2HTR1DHTR1BCHRM2DRD2
SCHEMBL7700411 0.87 CCR2 (0.51) CCR2HTR1DHTR1BCHRM2DRD2
SCHEMBL7702544 0.87 CCR2 (0.62) CCR2
SCHEMBL7702941 0.84 CCR2 (0.51) CCR2
SCHEMBL7702720 0.81 CCR2 (0.61) CCR2HTR1DHTR1BCHRM2DRD2
SCHEMBL7694620 0.81 CCR2 (0.56) CCR2HTR1DHTR1BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002079190-A1 3-SUBSTITUTED INDOLES AS CHEMOKINE ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-10-10 WO disclosed