SCHEMBL7702197

SCHEMBL7702197

CC(C)(C)OC(=O)N(Cc1ccc(F)cc1)S(C)(=O)=O

nearest known ligand 0.76

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 2/20 0.43
KCNA5 P22460 1/20 0.43
TAS2R14 Q9NYV8 5/20 0.43
KDM1A O60341 2/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
NR1D1 P20393 1/20 0.41
KCNQ4 P56696 1/20 0.41
KCNQ5 Q9NR82 1/20 0.41
GRM2 Q14416 1/20 0.40
PTGER2 P43116 2/20 0.40
YAP1 P46937 1/20 0.40
TEAD4 Q15561 1/20 0.40
TEAD2 Q15562 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705112 0.87 STAT5B (0.46) TAS2R14
SCHEMBL7707821 0.87 AKT1 (0.48) RIPK1
SCHEMBL7707801 0.86 KMT2A (0.43) HDAC6
SCHEMBL7705341 0.86 TSHR (0.40)
SCHEMBL6338886 0.86 TAS2R14 (0.42) TAS2R14NR1D1PTGER2
SCHEMBL5708152 0.82 TAS2R14 (0.58) TAS2R14
SCHEMBL7430459 0.79 RIPK1 (0.59) RIPK1KDM1AHDAC8HDAC6NR1D1
SCHEMBL30027626 0.79 TSHR (0.39) TAS2R14PTGER2
SCHEMBL17553442 0.78 RIPK1 (0.47) RIPK1KDM1AHDAC8HDAC6NR1D1
SCHEMBL2897902 0.77 HDAC3 (0.46) RIPK1KDM1AHDAC8HDAC6NR1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355665-B1 ANTIHISTAMINES, ANTIALLERGENS AND IRRITABLE BOWEL SYNDROME. JAMES BLACK FOUNDATION LIMITED (GB) 2002-03-12 US disclosed
WO-1999005114-A2 1H-4(5)-SUBSTITUTED IMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS HISTAMINE H3 RECEPTOR LIGANDS JAMES BLACK FOUNDATION LIMITED (GB) 1999-02-04 WO disclosed