SCHEMBL7702407

SCHEMBL7702407

CN(CCO)c1ccc(C2=NCCc3ccccc32)cn1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.40
TACR3 P29371 2/20 0.40
TRPV1 Q8NER1 4/20 0.37
POLB P06746 1/20 0.37
NOS3 P29474 1/20 0.36
NOS2 P35228 1/20 0.36
DGAT1 O75907 1/20 0.35
ALOX5AP P20292 1/20 0.35
MAPK10 P53779 2/20 0.34
MAOA P21397 1/20 0.34
HCAR3 P49019 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CFTR P13569 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705693 0.83 NOS3 (0.42) POLBNOS3NOS2MAPK10MAOA
SCHEMBL7702043 0.76 NOS3 (0.44) NOS3NOS2MAPK10MAOAKDM4E
SCHEMBL7702344 0.73 MAOA (0.47) NOS3NOS2MAPK10MAOACA1
SCHEMBL7697815 0.73 NOS3 (0.41) NOS3NOS2MAPK10MAOAKDM4E
SCHEMBL7698312 0.72 NOS3 (0.43) NOS3NOS2MAOAKDM4EALDH1A1
SCHEMBL13805616 0.70 NOS3 (0.49) POLBNOS3NOS2MAPK10MAOA
SCHEMBL30965936 0.70 CA1 (0.52) NOS3NOS2MAPK10MAOAKDM4E
SCHEMBL21063722 0.70 CA1 (0.52) NOS3NOS2MAPK10MAOAKDM4E
SCHEMBL7704878 0.69 CNR2 (0.47)
SCHEMBL12324101 0.69 POLB (0.45) TRPV1POLBDGAT1ALOX5APHCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed