SCHEMBL7705187

SCHEMBL7705187

CCOC(=O)N1CCN(CCc2ccccc2O)CC1

nearest known ligand 0.69

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
ALDH1A1 P00352 8/20 0.59
KDM4E B2RXH2 5/20 0.59
POLB P06746 1/20 0.59
HRH3 Q9Y5N1 1/20 0.57
KMT2A Q03164 3/20 0.53
MAPT P10636 2/20 0.53
MEN1 O00255 1/20 0.52
TSHR P16473 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10925979 0.78 ADORA3 (0.54) ALDH1A1KDM4EPOLBKMT2AMAPT
SCHEMBL9054221 0.77 L3MBTL1 (0.64) GAASMN1; SMN2ALDH1A1POLBKMT2A
SCHEMBL9819864 0.76 SIGMAR1 (0.69) GAASMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL5242857 0.75 ALDH1A1 (0.53) SMN1; SMN2ALDH1A1POLBKMT2AMAPT
SCHEMBL6044228 0.75 ALDH1A1 (0.49) GAAALDH1A1KDM4EPOLBKMT2A
SCHEMBL28312981 0.75 HRH1 (0.52) ALDH1A1KDM4EPOLB
SCHEMBL7224481 0.74 GAA (1.00) GAASMN1; SMN2ALDH1A1KDM4EKMT2A
SCHEMBL27678708 0.74 HRH3 (1.00) GAAALDH1A1KDM4EHRH3MAPT
SCHEMBL9513162 0.74 HRH2 (0.60) ALDH1A1KDM4EPOLBKMT2AMEN1
SCHEMBL10902416 0.73 HRH2 (0.67) SMN1; SMN2ALDH1A1KMT2AMAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242399-A1 $g(a)-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB S.A. (BE) 2002-09-25 EP disclosed
WO-2001046167-A1 α-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB, S.A. (BE) 2001-06-28 WO disclosed