SCHEMBL7705284

SCHEMBL7705284

CC(C)(c1nc(-c2ccccc2Cl)c(-c2cccc(CO)c2)s1)c1c(Cl)cc(Cl)cc1-n1ncc(=O)[nH]c1=O

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.34
ABCB11 O95342 1/20 0.34
CNR1 P21554 4/20 0.32
CNR2 P34972 4/20 0.32
DHODH Q02127 1/20 0.32
MAPK14 Q16539 2/20 0.31
ABL1 P00519 1/20 0.30
EGFR P00533 1/20 0.30
PDGFRB P09619 1/20 0.30
KIT P10721 1/20 0.30
FGFR1 P11362 1/20 0.30
SRC P12931 1/20 0.30
PDGFRA P16234 1/20 0.30
BTK Q06187 1/20 0.30
MAP2K4 P45985 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6459797 0.90 P2RX7 (0.39) P2RX7ABCB11DHODHMAP2K4
SCHEMBL7705288 0.82 P2RX7 (0.37) P2RX7ABCB11DHODHBTKMAP2K4
SCHEMBL7135587 0.78 P2RX7 (0.38) P2RX7ABCB11
SCHEMBL6462166 0.78 P2RX7 (0.38) P2RX7ABCB11
SCHEMBL6461284 0.77 P2RX7 (0.35) P2RX7ABCB11CNR1CNR2
SCHEMBL6461628 0.74 ADORA2A (0.38) P2RX7ABCB11BTK
SCHEMBL6459898 0.74 THRB (0.39) P2RX7ABCB11
SCHEMBL6462754 0.73 P2RX7 (0.41) P2RX7ABCB11
SCHEMBL6464512 0.73 P2RX7 (0.34) P2RX7ABCB11CNR1CNR2MAPK14
SCHEMBL6460365 0.73 P2RX7 (0.34) P2RX7ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020010177-A1 IL-5 inhibiting 6-azauracil derivatives JANSSEN CILAG S.A. (FR) 2002-01-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020010177-A1 IL-5 inhibiting 6-azauracil derivatives ALOX5, IL5, IL6ST P2RX7 880/4885ABCB11 2670/4885CNR1 237/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.