SCHEMBL7708428

SCHEMBL7708428

Nc1ncc(-c2ccc(F)cc2)c(=O)[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.51
ADORA1 P30542 1/20 0.43
TDO2 P48775 1/20 0.42
RAB9A P51151 2/20 0.40
MAP4K4 O95819 2/20 0.39
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
KMT2A Q03164 1/20 0.38
BRD4 O60885 1/20 0.38
XDH P47989 1/20 0.38
TYMS P04818 3/20 0.38
MAPK14 Q16539 2/20 0.38
USP7 Q93009 1/20 0.38
ERCC1 P07992 1/20 0.38
ERCC4 Q92889 1/20 0.38
MASP2 O00187 1/20 0.37
TYMP P19971 1/20 0.37
TNKS O95271 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
PARP2 Q9UGN5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7714691 0.84 DGAT1 (0.43) NOS1MEN1KMT2AXDHTYMS
SCHEMBL7708406 0.83 LTA4H (0.50) TDO2RAB9AMAP4K4MEN1NPC1
SCHEMBL11545985 0.82 MASP2 (0.56) NOS1XDHMASP2FGFR1
SCHEMBL14072020 0.76 MAP4K4 (0.43) NOS1ADORA1RAB9AMAP4K4NPC1
SCHEMBL8221175 0.74 MASP2 (0.66) NOS1TDO2MAPK14MASP2GSK3A
SCHEMBL7712456 0.72 MEN1 (0.44) NOS1MEN1KMT2AXDHTYMS
SCHEMBL11542411 0.71
SCHEMBL14081814 0.70 ESR1 (0.38) ADORA1MAPK14ABL1GSK3AGSK3B
SCHEMBL27552529 0.68 ADORA1 (0.49) NOS1ADORA1TDO2RAB9AMAP4K4
SCHEMBL12820646 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6440965-B1 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system KRENITSKY PHARMACEUTICALS, INC. 2002-08-27 US disclosed