SCHEMBL7708406

SCHEMBL7708406

Nc1ncc(-c2ccc(Cl)cc2)c(=O)[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.50
TRPV1 Q8NER1 1/20 0.46
MAP4K4 O95819 6/20 0.44
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 2/20 0.43
GAA P10253 2/20 0.43
RUNX1 Q01196 1/20 0.43
CBFB Q13951 1/20 0.43
TDO2 P48775 1/20 0.42
POLB P06746 1/20 0.42
XDH P47989 1/20 0.41
MAPT P10636 1/20 0.41
RECQL P46063 1/20 0.41
CYP1A2 P05177 1/20 0.41
KCNH2 Q12809 1/20 0.41
MINK1 Q8N4C8 1/20 0.41
TNIK Q9UKE5 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
RAB9A P51151 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7714691 0.84 DGAT1 (0.43) ALDH1A1GAAXDHMAPTMEN1
SCHEMBL7708428 0.83 NOS1 (0.51) MAP4K4TDO2XDHMEN1KMT2A
SCHEMBL11545985 0.82 MASP2 (0.56) ALDH1A1XDHMAPT
SCHEMBL6049622 0.79 TYMS (0.44) ALDH1A1KDM4EGAAMAPTMEN1
SCHEMBL19471383 0.74 LTA4H (0.81) LTA4HPOLBMAPTRAB9ANPC1
SCHEMBL5202998 0.72 LTA4H (0.57) LTA4HALDH1A1KDM4EXDHMAPT
SCHEMBL5206921 0.72 PLA2G7 (0.49) LTA4H
SCHEMBL6049582 0.72 NUDT1 (0.50) XDH
SCHEMBL7512558 0.72 RXFP1 (0.50) LTA4HALDH1A1KDM4EXDHCYP1A2
SCHEMBL2227162 0.71 KMO (0.54) MAP4K4XDHMINK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6440965-B1 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system KRENITSKY PHARMACEUTICALS, INC. 2002-08-27 US disclosed