SCHEMBL7708431

SCHEMBL7708431

CC(=O)Nc1cccc(-c2cc(N)n3nc(-c4ccno4)nc3c2)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
FYN P06241 9/20 0.41
CA2 P00918 1/20 0.41
HSD17B1 P14061 1/20 0.40
HSD17B2 P37059 1/20 0.40
NQO2 P16083 1/20 0.40
KDM4E B2RXH2 2/20 0.40
SYK P43405 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
MAP4K4 O95819 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
BACE1 P56817 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7484739 0.85 ADORA2A (0.52)
SCHEMBL7705969 0.85 MAPT (0.52) POLBTP53MAPTFYNHSD17B1
SCHEMBL7481934 0.85 ADORA2A (0.54) POLBTP53MAPTFYNHSD17B1
SCHEMBL7705893 0.82 ADORA2A (0.52) TP53MAPTFYNKDM4ERXFP1
SCHEMBL7708828 0.81 RAB9A (0.51) TP53MAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL7703234 0.81 ADORA2A (0.38) MAP4K4ALDH1A1SMN1; SMN2
SCHEMBL7711711 0.80 ALDH1A1 (0.44) TP53KDM4EALDH1A1SMN1; SMN2
SCHEMBL7708391 0.80 ADORA2A (0.45) MAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL7705871 0.80 FYN (0.55) TP53MAPTFYNNQO2KDM4E
SCHEMBL7705951 0.79 BACE1 (0.40) MAP4K4ALDH1A1SMN1; SMN2BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed