SCHEMBL7709280

SCHEMBL7709280

CC(C)(C)OC(=O)Nc1c(Br)ccc2ccc(OS(C)(=O)=O)cc12

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
NQO2 P16083 1/20 0.38
KAT6A Q92794 1/20 0.35
LCK P06239 4/20 0.35
CA1 P00915 6/20 0.35
CA2 P00918 6/20 0.35
CA12 O43570 5/20 0.35
CA9 Q16790 5/20 0.35
SMN1; SMN2 Q16637 1/20 0.33
ATR Q13535 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
GAA P10253 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
ACACB O00763 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7717601 0.84 ALDH1A1 (0.37) ALDH1A1NQO2KAT6ALCKCA1
SCHEMBL486679 0.81 ALDH1A1 (0.39) ALDH1A1CA1CA2CA12CA9
SCHEMBL7714050 0.81 CA12 (0.41) ALDH1A1NQO2LCKCA1CA12
SCHEMBL7717690 0.81 NQO2 (0.51) NQO2LCKCA1CA12CA9
SCHEMBL487112 0.80 TRPV1 (0.44) ALDH1A1NQO2KAT6ACA1CA2
SCHEMBL24150453 0.75 NQO2 (0.42) NQO2LCKCA1CA12CA9
SCHEMBL1530133 0.73 ENPP3 (0.52) ALDH1A1CA1CA2CA12CA9
SCHEMBL24150706 0.73 LCK (0.45) NQO2LCKCA1CA12CA9
SCHEMBL7714920 0.72 MEN1 (0.42) NQO2KAT6ACA1CA12NPSR1
SCHEMBL10062583 0.72 ALDH1A1 (0.39) ALDH1A1KAT6ACA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441017-B1 Inhibitors of prenyl-protein transferase MERCK & CO., INC. 2002-08-27 US disclosed
EP-1214326-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001018006-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed