SCHEMBL7709640

SCHEMBL7709640

CC(=O)Nc1c(O)c(C)c2c3c(cccc13)C(=O)OC2=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 5/20 0.40
ALDH1A1 P00352 5/20 0.39
POLB P06746 3/20 0.39
KDM4E B2RXH2 3/20 0.39
MAPT P10636 2/20 0.39
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
MAPK1 P28482 1/20 0.37
CASP1 P29466 1/20 0.37
CYP2C19 P33261 1/20 0.37
CASP7 P55210 1/20 0.37
USP2 O75604 2/20 0.36
BLM P54132 1/20 0.36
MAOA P21397 2/20 0.36
LMNA P02545 1/20 0.36
TNNI3 P19429 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7709792 0.84 KDM4E (0.49) TYMSALDH1A1POLBKDM4EMEN1
SCHEMBL7706686 0.74 TYMS (0.44) TYMSALDH1A1POLBKDM4EMEN1
SCHEMBL8319288 0.72 TDP2 (0.40) TYMSALDH1A1KDM4EMEN1KMT2A
SCHEMBL9079822 0.71 TYMS (0.46) TYMSALDH1A1POLBKDM4EMAPT
SCHEMBL7706770 0.71 KDM4E (0.63) TYMSALDH1A1KDM4EMAPTMEN1
SCHEMBL7703727 0.70 TYMS (0.45) TYMSPOLBKDM4EMAPTMEN1
SCHEMBL29860722 0.68 MAOA (0.61) ALDH1A1KDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL303302 0.68 MAOA (0.61) ALDH1A1KDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL15580925 0.68 MAOA (0.61) ALDH1A1KDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL8547705 0.68 TYMS (0.46) TYMSALDH1A1POLBKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed