SCHEMBL7709792

SCHEMBL7709792

COc1c(C)c2c3c(cccc3c1NC(C)=O)C(=O)OC2=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.49
CYP1A2 P05177 3/20 0.49
CYP2C9 P11712 3/20 0.49
IDO1 P14902 1/20 0.49
EGFR P00533 1/20 0.39
TYMS P04818 5/20 0.38
POLB P06746 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 3/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 2/20 0.35
MAPK1 P28482 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
ADORA3 P0DMS8 2/20 0.34
ADORA2A P29274 2/20 0.34
ADORA2B P29275 2/20 0.34
HSD17B10 Q99714 2/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319288 0.86 TDP2 (0.40) KDM4ECYP1A2CYP2C9IDO1EGFR
SCHEMBL7709640 0.84 TYMS (0.40) KDM4ECYP1A2CYP2C9TYMSPOLB
SCHEMBL7706686 0.71 TYMS (0.44) KDM4ECYP1A2CYP2C9TYMSPOLB
SCHEMBL9079822 0.69 TYMS (0.46) KDM4ECYP1A2TYMSPOLBMEN1
SCHEMBL7706770 0.68 KDM4E (0.63) KDM4ETYMSMEN1KMT2AALDH1A1
SCHEMBL7703727 0.68 TYMS (0.45) KDM4ECYP1A2CYP2C9TYMSPOLB
SCHEMBL8547705 0.66 TYMS (0.46) KDM4ECYP1A2CYP2C9TYMSPOLB
SCHEMBL15580925 0.66 MAOA (0.61) KDM4ECYP1A2CYP2C9ALDH1A1CYP3A4
SCHEMBL29860722 0.66 MAOA (0.61) KDM4ECYP1A2CYP2C9ALDH1A1CYP3A4
SCHEMBL303302 0.66 MAOA (0.61) KDM4ECYP1A2CYP2C9ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed