SCHEMBL7711245

SCHEMBL7711245

CC1=C(N)Nc2cc(C(N)(Cc3cccc(F)c3)C(=O)OC(C)(C)C)ccc2O1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 1/20 0.33
LTB4R2 Q9NPC1 1/20 0.33
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
TSHR P16473 2/20 0.31
LMNA P02545 1/20 0.31
PPARG P37231 1/20 0.31
NCOA2 Q15596 1/20 0.31
NCOA1 Q15788 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31
CHRM1 P11229 1/20 0.30
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
RIPK1 Q13546 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7711358 0.90 ACE2 (0.34) ALDH1A1NPSR1
SCHEMBL7708351 0.90
SCHEMBL7704909 0.90 MMP8 (0.31) LTB4RLTB4R2SMN1; SMN2
SCHEMBL7704899 0.89 PKM (0.35) POLBSMN1; SMN2RIPK1
SCHEMBL7704869 0.89 GRM2 (0.33) CTSKLMNACHRM1ALDH1A1
SCHEMBL7711363 0.87 EPHX2 (0.30)
SCHEMBL7711183 0.86 NR3C2 (0.40) TSHRLMNAALDH1A1POLBSMN1; SMN2
SCHEMBL7708186 0.86
SCHEMBL7710866 0.85 KDM4E (0.31) ALDH1A1
SCHEMBL7711454 0.85 FDPS (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed