SCHEMBL7704869

SCHEMBL7704869

COc1cccc(CC(N)(C(=O)OC(C)(C)C)c2ccc3c(c2)NC(N)=C(C)O3)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.33
GRM3 Q14832 1/20 0.33
TP53 P04637 1/20 0.33
ALDH1A1 P00352 4/20 0.33
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
MAPT P10636 2/20 0.33
CTSK P43235 1/20 0.33
PTPRB P23467 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
ALOX15 P16050 1/20 0.33
GFER P55789 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CHRM1 P11229 1/20 0.33
CTBP2 P56545 1/20 0.32
RAB9A P51151 1/20 0.32
KDM4E B2RXH2 1/20 0.32
USP2 O75604 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7704944 0.90 ALDH1A1 (0.32) ALDH1A1MEN1KMT2AMAPTHSD17B10
SCHEMBL7704899 0.89 PKM (0.35) KDM4E
SCHEMBL7711245 0.89 LTB4R (0.33) ALDH1A1CTSKLMNACHRM1
SCHEMBL7711358 0.88 ACE2 (0.34) GRM2GRM3ALDH1A1MAPTGAA
SCHEMBL7711183 0.87 NR3C2 (0.40) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL7711363 0.86 EPHX2 (0.30)
SCHEMBL7711454 0.84 FDPS (0.32)
SCHEMBL7704963 0.84 CYP3A4 (0.34) LMNAGAA
SCHEMBL7708351 0.84
SCHEMBL7711304 0.83 CYP3A4 (0.36) TP53ALDH1A1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed