SCHEMBL7712435

SCHEMBL7712435

O=C(Cn1nc(S(=O)(=O)Cc2ccc(F)cc2)c2ccc(F)cc21)N(Cc1ccc(F)cc1)C1CC1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 4/20 0.48
HCRTR1 O43613 4/20 0.48
OPRM1 P35372 3/20 0.38
TMEM97 Q5BJF2 2/20 0.38
CFD P00746 3/20 0.38
TACR1 P25103 1/20 0.38
NSD2 O96028 1/20 0.37
HTR2A P28223 3/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
GAA P10253 1/20 0.35
PER2 O15055 1/20 0.35
CRY1 Q16526 1/20 0.35
CRY2 Q49AN0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7711206 0.96 HCRTR2 (0.55) HCRTR2HCRTR1OPRM1TMEM97CFD
SCHEMBL7707039 0.94 HCRTR2 (0.47) HCRTR2HCRTR1OPRM1TMEM97CFD
SCHEMBL7702319 0.81 HCRTR2 (0.47) HCRTR2HCRTR1PTGDR2
SCHEMBL2592050 0.81 THRB (0.46) HCRTR2HCRTR1
SCHEMBL7702650 0.79 HCRTR2 (0.78) HCRTR2HCRTR1
SCHEMBL7709100 0.77 SMN1; SMN2 (0.51) HCRTR2HCRTR1GAA
SCHEMBL2588992 0.77 HCRTR2 (0.44) HCRTR2HCRTR1
SCHEMBL7713631 0.76 HCRTR2 (0.61) HCRTR2HCRTR1
SCHEMBL7713640 0.75 HCRTR2 (0.54) HCRTR2HCRTR1PTGDR2
SCHEMBL2594744 0.75 HCRTR1 (0.48) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011138265-A2 INDOLE AND INDAZOLE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS EVOTEC AG (DE) 2011-11-10 WO disclosed