SCHEMBL7714689

SCHEMBL7714689

COC1(OC)[N]C=Cc2ccccc21

nearest known ligand 0.31

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18403739 0.64 OXTR (0.32) KDM4EPKM
SCHEMBL5136349 0.63 GAA (0.32) KDM4EPKM
SCHEMBL11034491 0.60 KDM4E (0.36) KDM4EPKM
SCHEMBL5837474 0.60 KDM4E (0.39) KDM4EPKM
SCHEMBL27390499 0.60 KDM4E (0.46) KDM4EPKM
SCHEMBL31756888 0.59 KDM4E (0.35) KDM4EPKM
SCHEMBL8429771 0.59 KDM4E (0.35) KDM4EPKM
SCHEMBL6545109 0.59 KDM4E (0.35) KDM4EPKM
SCHEMBL9666306 0.59 KDM4E (0.38) KDM4EPKM
SCHEMBL13105950 0.58 MAPT (0.33) KDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191142-B1 Aroyl aminoacyl pyrroles for use in the treatment of neuropathic pain ORTHO-MCNEIL PHARMACEUTICAL, INC. 2001-02-20 US claimed
US-6369228-B2 ANTICONVULSANTS ORTHO-MCNEIL PHARMACEUTICAL, INC. 2002-04-09 US disclosed
EP-1154996-A2 AROYL AMINOACYL PYRROLES FOR USE IN THE TREATMENT OF NEUROPATHIC PAIN Ortho-McNeil Pharmaceutical, Inc. (US) 2001-11-21 EP disclosed
US-6191142-B1 Aroyl aminoacyl pyrroles for use in the treatment of neuropathic pain ORTHO-MCNEIL PHARMACEUTICAL, INC. 2001-02-20 US disclosed
WO-2000048584-A2 AROYL AMINOACYL PYRROLES FOR USE IN THE TREATMENT OF NEUROPATHIC PAIN ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2000-08-24 WO disclosed