SCHEMBL7716692

SCHEMBL7716692

COc1ccc(CCc2cnc(N)[nH]c2=O)cc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
QTRT1 Q9BXR0 1/20 0.52
DAO P14920 3/20 0.48
CSF1R P07333 1/20 0.46
NTRK2 Q16620 1/20 0.46
ABL1 P00519 1/20 0.46
RIN1 Q13671 1/20 0.46
PLA2G7 Q13093 1/20 0.45
DHODH Q02127 1/20 0.44
TYMS P04818 1/20 0.44
TAAR1 Q96RJ0 1/20 0.42
XDH P47989 1/20 0.41
FABP4 P15090 1/20 0.41
ABCB1 P08183 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7716578 0.87 PLA2G7 (0.48) QTRT1PLA2G7TYMSXDH
SCHEMBL7716580 0.81 DAO (0.50) DAOPLA2G7TYMSTAAR1XDH
SCHEMBL8239236 0.80 BACE1 (0.53) DAODHODHABCB1
SCHEMBL7712501 0.74 XDH (0.45) TYMSXDH
SCHEMBL7708037 0.72 AOC3 (0.51) DAOPLA2G7
SCHEMBL13039021 0.71 NOS1 (0.42) TYMS
SCHEMBL5202767 0.71 PDE3B (0.47) DAOPLA2G7XDH
SCHEMBL4211345 0.71 TK1 (0.36) TYMS
SCHEMBL834551 0.69 TAAR1 (0.73) TAAR1
SCHEMBL10736648 0.69 PLA2G7 (0.49) DAOPLA2G7FABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6440965-B1 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system KRENITSKY PHARMACEUTICALS, INC. 2002-08-27 US disclosed