SCHEMBL7717820

SCHEMBL7717820

CC(C)(C)[Si](Oc1cccc2c1CCCC(=O)C2)(c1ccccc1)c1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RXRA P19793 7/20 0.33
RXRB P28702 7/20 0.33
RXRG P48443 4/20 0.33
P2RX7 Q99572 2/20 0.33
CYP2A6 P11509 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.31
DRD2 P14416 1/20 0.31
DRD1 P21728 1/20 0.31
DRD5 P21918 1/20 0.31
DRD3 P35462 1/20 0.31
SSTR4 P31391 1/20 0.31
BACE1 P56817 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7483555 0.93 CYP2A6 (0.38) CYP2A6BACE1
SCHEMBL7487183 0.80 ADRB2 (0.46) CYP2A6MRGPRX4
SCHEMBL2061100 0.75 DRD2 (0.47) DRD2DRD1DRD5DRD3
SCHEMBL8078287 0.75 DRD2 (0.37) DRD2DRD3
SCHEMBL7718293 0.74
SCHEMBL5153891 0.74 ADRB2 (0.37) MRGPRX4BACE1
SCHEMBL7718298 0.74 TRPA1 (0.32)
SCHEMBL7713227 0.74 CYP19A1 (0.37) DRD2
SCHEMBL7718886 0.74 MTNR1A (0.39) DRD2DRD3SSTR4
SCHEMBL7486376 0.73 DRD2 (0.58) DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6384072-B1 CARBAMYL SUBSTITUTED COMPOUNDS WITH ETHER GROUPS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-05-07 US disclosed
EP-1030834-A1 BENZOCYCLOHEPTENE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-30 EP disclosed
WO-1999024397-A1 BENZOCYCLOHEPTENE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-05-20 WO disclosed