SCHEMBL7718684

SCHEMBL7718684

CCc1c(N2CCCCC2)cc2c(c1OC)C(=O)NC2=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 5/20 0.41
CDK4 P11802 3/20 0.41
CCND1 P24385 3/20 0.41
CDK2 P24941 3/20 0.35
CCNA2 P20248 1/20 0.35
CCNA1 P78396 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MAPT P10636 2/20 0.34
TNNI3 P19429 1/20 0.34
TNNT2 P45379 1/20 0.34
TNNC1 P63316 1/20 0.34
HTR1A P08908 2/20 0.34
DRD2 P14416 2/20 0.34
DRD4 P21917 2/20 0.34
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
DRD3 P35462 2/20 0.34
KDR P35968 2/20 0.32
FLT3 P36888 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7722008 0.80 CDK4 (0.35) GSK3BCDK4CCND1MEN1KMT2A
SCHEMBL7723028 0.80 CDK4 (0.35) GSK3BCDK4CCND1MEN1KMT2A
SCHEMBL5996608 0.76 PARP1 (0.39) MEN1KMT2AMAPTALDH1A1ALDH1A3
Hydrochloric Acid SCHEMBL7723748 0.75 PARP1 (0.38) GSK3BMEN1KMT2AMAPTALDH1A1
Hydrochloric Acid SCHEMBL8347114 0.72 HTR2C (0.51) DRD2HTR2AHTR2CDRD3ACHE
SCHEMBL7883990 0.69 HTR1A (0.38) GSK3BCDK4CCND1HTR1ADRD2
SCHEMBL7964016 0.68 KMT2A (0.36) MEN1KMT2AMAPTALDH1A1ALDH1A3
SCHEMBL29614674 0.66 PARP1 (0.43) GSK3BCDK4CCND1MEN1KMT2A
SCHEMBL7722975 0.66 HTR1A (0.43) HTR1ADRD2DRD4HTR2AHTR2C
Hydrochloric Acid SCHEMBL7727011 0.66 KDM4E (0.43) MEN1KMT2AMAPTALDH1A1ALDH1A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37729-E1 4-Heteroaryl-1-piperidinealkylamines and derivatives thereof and their therapeutic utility AVENTIS PHARMACEUTICALS INC. 2002-06-04 US disclosed
US-RE37478-E1 COMPOUNDS WITH HETEROCYCLIC AMINO COMPOUNDS AVENTIS PHARMACEUTICALS, INC. 2001-12-18 US disclosed
US-RE37029-E1 ANTIPSYCHOTIC AND ANALGESIC AGENTS AVENTIS PHARMACEUTICALS INC. 2001-01-23 US disclosed