SCHEMBL7722008

SCHEMBL7722008

CCc1c(N)c(N2CCCCC2)cc2c1C(=O)NC2=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
GSK3B P49841 1/20 0.35
CASP3 P42574 2/20 0.33
TERT O14746 1/20 0.33
CASP2 P42575 1/20 0.33
CASP7 P55210 1/20 0.33
CASP6 P55212 1/20 0.33
CASP8 Q14790 1/20 0.33
ALDH1A1 P00352 5/20 0.33
KDM4E B2RXH2 4/20 0.33
HTT P42858 3/20 0.33
LMNA P02545 2/20 0.33
L3MBTL1 Q9Y468 3/20 0.31
GAA P10253 3/20 0.31
S100B P04271 2/20 0.31
MEN1 O00255 2/20 0.31
MAPK1 P28482 2/20 0.31
KMT2A Q03164 2/20 0.31
MAPT P10636 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7723028 0.84 CDK4 (0.35) CDK4CCND1GSK3BCASP3CASP2
SCHEMBL5996608 0.81 PARP1 (0.39) ALDH1A1HTTLMNAL3MBTL1GAA
Hydrochloric Acid SCHEMBL7723748 0.80 PARP1 (0.38) GSK3BALDH1A1KDM4EHTTLMNA
SCHEMBL7718684 0.80 GSK3B (0.41) CDK4CCND1GSK3BALDH1A1MEN1
SCHEMBL7883990 0.74 HTR1A (0.38) CDK4CCND1GSK3BALDH1A1
SCHEMBL7722975 0.70 HTR1A (0.43)
Hydrochloric Acid SCHEMBL7727011 0.70 KDM4E (0.43) ALDH1A1KDM4EHTTLMNAL3MBTL1
Hydrochloric Acid SCHEMBL7882760 0.69 HTR1A (0.42) LMNAMAPT
SCHEMBL7964016 0.69 KMT2A (0.36) ALDH1A1KDM4EHTTLMNAL3MBTL1
SCHEMBL29614674 0.68 PARP1 (0.43) CDK4CCND1GSK3BCASP3CASP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37729-E1 4-Heteroaryl-1-piperidinealkylamines and derivatives thereof and their therapeutic utility AVENTIS PHARMACEUTICALS INC. 2002-06-04 US disclosed
US-RE37478-E1 COMPOUNDS WITH HETEROCYCLIC AMINO COMPOUNDS AVENTIS PHARMACEUTICALS, INC. 2001-12-18 US disclosed