SCHEMBL7723028

SCHEMBL7723028

CCc1c(O)c(N2CCCCC2)cc2c1C(=O)NC2=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
GSK3B P49841 1/20 0.35
ALDH1A1 P00352 5/20 0.33
MAPT P10636 4/20 0.33
HPGD P15428 3/20 0.33
TSHR P16473 1/20 0.33
CASP3 P42574 2/20 0.33
CASP2 P42575 1/20 0.33
CASP7 P55210 1/20 0.33
CASP6 P55212 1/20 0.33
CASP8 Q14790 1/20 0.33
RAB9A P51151 4/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
NPC1 O15118 2/20 0.32
WEE1 P30291 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
LIPE Q05469 1/20 0.32
GAA P10253 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7722008 0.84 CDK4 (0.35) CDK4CCND1GSK3BALDH1A1MAPT
SCHEMBL5996608 0.81 PARP1 (0.39) ALDH1A1MAPTHPGDTSHRRAB9A
Hydrochloric Acid SCHEMBL7723748 0.80 PARP1 (0.38) GSK3BALDH1A1MAPTHPGDTSHR
SCHEMBL7718684 0.80 GSK3B (0.41) CDK4CCND1GSK3BALDH1A1MAPT
SCHEMBL7883990 0.74 HTR1A (0.38) CDK4CCND1GSK3BALDH1A1
SCHEMBL8350209 0.71 HTR2C (0.53) ACHE
SCHEMBL7722975 0.70 HTR1A (0.43)
Hydrochloric Acid SCHEMBL7727011 0.70 KDM4E (0.43) ALDH1A1MAPTHPGDTSHRRAB9A
Hydrochloric Acid SCHEMBL7882760 0.69 HTR1A (0.42) MAPTLMNA
SCHEMBL7964016 0.69 KMT2A (0.36) ALDH1A1MAPTHPGDTSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37729-E1 4-Heteroaryl-1-piperidinealkylamines and derivatives thereof and their therapeutic utility AVENTIS PHARMACEUTICALS INC. 2002-06-04 US disclosed
US-RE37478-E1 COMPOUNDS WITH HETEROCYCLIC AMINO COMPOUNDS AVENTIS PHARMACEUTICALS, INC. 2001-12-18 US disclosed
US-RE37029-E1 ANTIPSYCHOTIC AND ANALGESIC AGENTS AVENTIS PHARMACEUTICALS INC. 2001-01-23 US disclosed