SCHEMBL7723172

SCHEMBL7723172

O=C(NC1CCN(CCc2ccc(F)cc2)C1)C(c1cccs1)c1cccs1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.52
DRD4 P21917 4/20 0.52
DRD2 P14416 3/20 0.52
CHRM2 P08172 1/20 0.49
CHRM1 P11229 1/20 0.49
CHRM3 P20309 1/20 0.49
HTR2C P28335 2/20 0.45
HTR7 P34969 2/20 0.45
HTR6 P50406 1/20 0.45
TSHR P16473 1/20 0.43
SIGMAR1 Q99720 3/20 0.42
CCR3 P51677 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7723166 1.00 HTR2A (0.52) HTR2ADRD4DRD2CHRM2CHRM1
SCHEMBL7729407 0.81 SIGMAR1 (0.48) HTR2ADRD4DRD2HTR2CHTR7
SCHEMBL7729412 0.81 SIGMAR1 (0.48) HTR2ADRD4DRD2HTR2CHTR7
SCHEMBL7724234 0.80 DRD2 (0.45) HTR2ADRD4DRD2HTR2CHTR7
SCHEMBL7724237 0.80 DRD2 (0.45) HTR2ADRD4DRD2HTR2CHTR7
SCHEMBL7729521 0.79 DRD2 (0.45) HTR2ADRD4DRD2HTR2CHTR7
SCHEMBL7729514 0.79 DRD2 (0.45) HTR2ADRD4DRD2HTR2CHTR7
SCHEMBL7724283 0.78 CCR3 (0.50) HTR2ADRD4DRD2HTR2CHTR7
SCHEMBL7724290 0.78 CCR3 (0.50) HTR2ADRD4DRD2HTR2CHTR7
SCHEMBL7729558 0.74 CCR1 (0.60) HTR2ADRD4CHRM3HTR2CTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6468998-B1 ANTAGONIZE SEROTONIN 2 RECEPTORS, SUPPRESS PLATELET AGGREGATION, IMPROVE PERIPHERAL CIRCULATION AND PROMOTE LACHRYMATION MITSUBISHI PHARMA CORPORATION (JP) 2002-10-22 US disclosed
EP-1125922-A1 PYRROLIDINE COMPOUNDS AND MEDICINAL UTILIZATION THEREOF Welfide Corporation (JP) 2001-08-22 EP disclosed