SCHEMBL7728708

SCHEMBL7728708

O=C(N[C@H](CCc1ccccc1)C(=O)Oc1c(F)c(F)c(F)c(F)c1F)OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSL P07711 12/20 0.55
CTSK P43235 6/20 0.52
CTSB P07858 4/20 0.49
CTSS P25774 2/20 0.49
CASP1 P29466 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7333168 0.88 CTSK (0.59) CTSLCTSKCTSBCTSS
SCHEMBL7333172 0.88 CTSK (0.59) CTSLCTSKCTSBCTSS
SCHEMBL2066047 0.88 CTSK (0.54) CTSLCTSKCTSBCTSS
SCHEMBL27857319 0.87 CA1 (0.53) CTSLCTSKCTSBCTSS
SCHEMBL16494692 0.86 SIRT2 (0.53) CTSLCTSKCTSS
SCHEMBL16494690 0.86 SIRT2 (0.53) CTSLCTSKCTSS
SCHEMBL7302369 0.84 PSMB1 (0.55) CTSLCTSKCTSBCTSSCASP1
SCHEMBL27616333 0.83 CTSL (0.61) CTSLCTSKCTSBCTSSCASP1
SCHEMBL6139194 0.83 CTSL (0.61) CTSLCTSKCTSBCTSSCASP1
SCHEMBL2367306 0.82 CTSK (0.67) CTSLCTSKCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed
WO-2000001714-A1 EFFLUX PUMP INHIBITORS MICROCIDE PHARMACEUTICALS, INC. (US) 2000-01-13 WO disclosed