SCHEMBL7728745

SCHEMBL7728745

CC(C)(C)OC(=O)N1C[C@H](N(C(=O)CN)C(=O)OC(C)(C)C)C[C@H]1C(=O)N1CCN(c2cccc(Cl)c2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.44
LMNA P02545 4/20 0.43
TSHR P16473 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ALDH1A1 P00352 4/20 0.41
CPT2 P23786 1/20 0.41
CPT1A P50416 1/20 0.41
NR1H2 P55055 1/20 0.41
NR1H3 Q13133 1/20 0.41
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
TGM2 P21980 1/20 0.40
HTR1A P08908 1/20 0.40
HTR2A P28223 1/20 0.40
HTR7 P34969 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7730697 0.91 SMN1; SMN2 (0.44) MAPTLMNATSHRALDH1A1KMT2A
SCHEMBL7722004 0.87 TGM2 (0.40) MAPTLMNAKMT2AMEN1TGM2
SCHEMBL7734014 0.86 GAA (0.40) MAPTLMNACYP1A2CYP3A4CYP2D6
SCHEMBL7722244 0.80 GPR119 (0.36)
SCHEMBL7722094 0.80 GPR119 (0.36)
SCHEMBL7727837 0.78 SIGMAR1 (0.43)
SCHEMBL7728662 0.77 DPP4 (0.42) KMT2AMEN1TGM2HTR1AHTR2A
SCHEMBL7730641 0.77 NPBWR1 (0.39) LMNACYP1A2CYP3A4CYP2C19NPSR1
SCHEMBL7722097 0.77 TGM2 (0.39) MAPTLMNAALDH1A1TGM2HTR2A
SCHEMBL7728192 0.75 POLB (0.47) CYP1A2CYP3A4CYP2C19ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed
WO-2000001714-A1 EFFLUX PUMP INHIBITORS MICROCIDE PHARMACEUTICALS, INC. (US) 2000-01-13 WO disclosed