SCHEMBL7732369

SCHEMBL7732369

NC[C@@H](N)C(=O)N[C@H](CCc1ccccc1)c1nc(C(=O)Nc2cnc3cc(OC(=O)C(F)(F)F)ccc3c2)co1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
MAPT P10636 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
SRC P12931 3/20 0.33
ZAP70 P43403 3/20 0.33
SCN9A Q15858 1/20 0.32
TRPV1 Q8NER1 6/20 0.32
HPGDS O60760 1/20 0.32
ROCK2 O75116 2/20 0.31
KDR P35968 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7735549 0.88 LTA4H (0.38) NPC1RAB9AMAPTNFKB1NFKB2
Trifluoroacetic Acid SCHEMBL7723297 0.82 RAB9A (0.41) NPC1RAB9AMAPTNFKB1NFKB2
SCHEMBL7735983 0.80 RAB9A (0.44) NPC1RAB9AMAPTNFKB1NFKB2
SCHEMBL7730721 0.75 LTA4H (0.40) NPC1RAB9AMAPTSMN1; SMN2SRC
SCHEMBL7723198 0.75 TRPV1 (0.38) NPC1RAB9AMAPTNFKB1NFKB2
Trifluoroacetic Acid SCHEMBL7735917 0.75 RAB9A (0.48) NPC1RAB9AMAPTNFKB1NFKB2
SCHEMBL7733896 0.75 RAB9A (0.38) NPC1RAB9AMAPTNFKB1NFKB2
SCHEMBL7732103 0.72 RAB9A (0.53) NPC1RAB9AMAPTNFKB1NFKB2
Trifluoroacetic Acid SCHEMBL7733887 0.72 RAB9A (0.39) NPC1RAB9AMAPTNFKB1NFKB2
SCHEMBL7733986 0.72 PSMD14 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436980-B1 TRANSPORT PROTEIN SUPPRESSORS; MICROBIOCIDES ESSENTIAL THERAPEUTICS, INC. 2002-08-20 US disclosed
US-6204279-B1 SECONDARY AMIDE CONTAINING BENZOXAZOLE DERIVATIVES MICROCIDE PHARMACEUTICALS, INC. 2001-03-20 US disclosed