SCHEMBL7733863

SCHEMBL7733863

CC(C)(C)[Si](C)(C)OCCCc1c[nH]c2ccc(F)cc12

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MPO P05164 17/20 0.56
SLC6A4 P31645 4/20 0.56
HTR2A P28223 1/20 0.52
TRPM8 Q7Z2W7 1/20 0.52
HTR1A P08908 2/20 0.52
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8140362 0.93 MPO (0.55) MPOSLC6A4HTR2ATRPM8HTR1A
SCHEMBL22152521 0.85 SLC6A4 (0.56) SLC6A4HTR2ATRPM8HTR1A
SCHEMBL8129433 0.82 HTR2A (0.55) MPOSLC6A4HTR2ATRPM8HTR1A
SCHEMBL5946187 0.82 SLC6A4 (0.52) MPOSLC6A4HTR2AHTR1AKMT2A
SCHEMBL1304576 0.79 MPO (0.60) MPOSLC6A4HTR2ATRPM8HTR1A
SCHEMBL14499878 0.79 MPO (0.60) MPOSLC6A4HTR2ATRPM8
SCHEMBL9093555 0.78 HTR2A (0.55) SLC6A4HTR2ATRPM8HTR1A
SCHEMBL28604379 0.76 HTR1A (0.34) MPOSLC6A4HTR2ATRPM8HTR1A
SCHEMBL27561383 0.76 MPO (0.79) MPOSLC6A4HTR2ATRPM8
SCHEMBL30817963 0.76 DUT (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6828325-B2 A benzoxazolopiperazine derivative useful for treating Parkinson's diseases, schizophrenia, anxiety and depression SOLVAY PHARMACEUTICALS B.V. (CH) 2004-12-07 US disclosed