SCHEMBL7734332

SCHEMBL7734332

CC(C)Nc1nc2cc(C#N)ccc2n1[C@@H]1O[C@H](C)[C@@H](O)[C@H]1O

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.50
IDH1 O75874 10/20 0.42
TRPV4 Q9HBA0 2/20 0.41
ADK P55263 2/20 0.37
HSPA8 P11142 1/20 0.35
GPR6 P46095 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7733484 0.93 HDAC6 (0.49) HDAC6IDH1TRPV4ADKHSPA8
SCHEMBL7734525 0.85 HDAC6 (0.57) HDAC6TRPV4ADKHSPA8
SCHEMBL7734310 0.83 HDAC6 (0.50) HDAC6IDH1ADKHSPA8
SCHEMBL7114052 0.82 HDAC6 (0.49) HDAC6IDH1TRPV4HSPA8
SCHEMBL7734315 0.81 TRPV4 (0.38) HDAC6IDH1TRPV4GPR6
SCHEMBL7118656 0.81 HDAC6 (0.48) HDAC6IDH1TRPV4ADK
SCHEMBL7215020 0.80 HDAC6 (0.74) HDAC6TRPV4ADKHSPA8
SCHEMBL7738034 0.80 HDAC6 (0.56) HDAC6HSPA8
SCHEMBL10308324 0.80 HDAC6 (0.74) HDAC6TRPV4ADKHSPA8
SCHEMBL7215024 0.80 HDAC6 (0.74) HDAC6TRPV4ADKHSPA8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6413938-B1 HERPES VIRUS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2002-07-02 US disclosed
EP-0970100-A1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 2000-01-12 EP disclosed
WO-1998035977-A1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 1998-08-20 WO disclosed