SCHEMBL7118656

SCHEMBL7118656

CC(C)Nc1nc2cc([N+](=O)[O-])ccc2n1[C@@H]1O[C@H](C)[C@@H](O)[C@H]1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.48
SLC29A1 Q99808 1/20 0.38
TRPV4 Q9HBA0 1/20 0.38
IRAK4 Q9NWZ3 5/20 0.38
PKM P14618 2/20 0.36
ALDH1A1 P00352 3/20 0.36
MAPT P10636 3/20 0.36
LMNA P02545 2/20 0.35
MEN1 O00255 1/20 0.35
CYP2D6 P10635 1/20 0.35
KMT2A Q03164 1/20 0.35
ADK P55263 1/20 0.35
IDH1 O75874 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34
MAP3K7 O43318 1/20 0.34
IRAK1 P51617 1/20 0.34
KCNH3 Q9ULD8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7117206 0.93 HDAC6 (0.48) HDAC6SLC29A1TRPV4IRAK4ALDH1A1
SCHEMBL7120051 0.83 TRPV4 (0.38) HDAC6TRPV4IRAK4PKMALDH1A1
SCHEMBL7734525 0.82 HDAC6 (0.57) HDAC6TRPV4MAPTMEN1KMT2A
SCHEMBL7734310 0.81 HDAC6 (0.50) HDAC6PKMALDH1A1MEN1KMT2A
SCHEMBL7114052 0.80 HDAC6 (0.49) HDAC6TRPV4PKMMEN1KMT2A
SCHEMBL7215020 0.78 HDAC6 (0.74) HDAC6TRPV4ADK
SCHEMBL7738034 0.78 HDAC6 (0.56) HDAC6MAPTLMNASMN1; SMN2
SCHEMBL7215024 0.78 HDAC6 (0.74) HDAC6TRPV4ADK
SCHEMBL7742258 0.76 HDAC6 (0.57) HDAC6ALDH1A1MAPTMEN1KMT2A
SCHEMBL7733484 0.76 HDAC6 (0.49) HDAC6TRPV4ADKIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970100-B1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LTD (GB) 2003-11-12 EP claimed
US-6413938-B1 HERPES VIRUS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2002-07-02 US claimed
EP-0970100-B1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LTD (GB) 2003-11-12 EP disclosed
US-6413938-B1 HERPES VIRUS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2002-07-02 US disclosed
EP-0970100-A1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 2000-01-12 EP disclosed
WO-1998035977-A1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 1998-08-20 WO disclosed