SCHEMBL7737658

SCHEMBL7737658

OCCN1CCCCc2c(O)cccc21

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BCL2L1 Q07817 1/20 0.43
BAD Q92934 1/20 0.43
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
DRD2 P14416 4/20 0.37
HTR1A P08908 3/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
ADRA1B P35368 1/20 0.36
DRD1 P21728 1/20 0.36
DRD5 P21918 1/20 0.36
DRD3 P35462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8493200 0.89 MEN1 (0.42) DRD2HTR1ADRD1DRD5DRD3
SCHEMBL8497315 0.79 ALDH1A1 (0.40) DRD2HTR1AADRA1BDRD1DRD5
SCHEMBL4703874 0.79 NPC1 (0.41) BCL2L1BADHTR2CHTR2BHRH3
SCHEMBL14202152 0.78 KDM4E (0.55) CHRM2CHRM4CHRM1CHRM3
SCHEMBL22129196 0.78 HRH3 (0.51) BCL2L1BADHRH3DRD2HTR1A
SCHEMBL2743854 0.75 ADRA1B (0.42) BCL2L1BADHTR2CHTR2BHRH3
SCHEMBL7737082 0.74 HRH3 (0.46) HRH3HDAC1HDAC6
SCHEMBL15787244 0.74 DRD2 (0.47) DRD2HTR1ADRD1
SCHEMBL4701898 0.72 NOTUM (0.44) HRH3CHRM2CHRM4CHRM1CHRM3
SCHEMBL13911374 0.71 BCL2L1 (0.46) BCL2L1BADDRD2DRD1DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407096-B1 1,4-BENZOTHIAZINE AND 1,4-BENZOXAZINE DERIVATIVES; HYPOTENSIVE, ANTIISCHEMIC, ANTIALLERGEN, ANTIASTHMATIC AND ANTICOAGULANT AGENTS; CARDIOVASCULAR DISORDERS TORAY INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1028113-A1 FUSED BENZENE HETEROCYCLE DERIVATIVES AND UTILIZATION THEREOF TORAY INDUSTRIES, INC. (JP) 2000-08-16 EP disclosed