SCHEMBL7739889

SCHEMBL7739889

CCOP(=O)(OCC)c1cc2cc(-c3ccc(C(F)(F)F)cc3)c(F)cc2[nH]c1=O

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.35
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35
RAB9A P51151 1/20 0.34
MAOB P27338 1/20 0.34
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
TYMS P04818 1/20 0.33
SCN9A Q15858 2/20 0.32
KIF11 P52732 1/20 0.32
PDE2A O00408 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7740617 0.89 PTGES (0.36) CDK5CDK5R1RAB9AMAOBTYMS
SCHEMBL7742769 0.82 APP (0.39) APPCDK5CDK5R1AKR1C3AKR1C2
SCHEMBL6929177 0.82 CDK5 (0.39) CDK5CDK5R1KIF11
SCHEMBL7739895 0.81 AKR1C3 (0.36) APPCDK5CDK5R1RAB9AAKR1C3
SCHEMBL7735087 0.80 NTRK1 (0.35) RAB9A
SCHEMBL7739643 0.79 GSK3B (0.37)
Nitrogen SCHEMBL27548156 0.77 CDK5 (0.36) CDK5CDK5R1
SCHEMBL6928596 0.76 GRIN2D (0.33)
SCHEMBL6928527 0.76 PARP1 (0.40)
SCHEMBL7741117 0.75 PRKAG1 (0.37) RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420386-B1 SPINAL TRAUMATISM, EPILEPSY, CHRONIC NEURODEGENERATIVE DISEASES SUCH AS ALZHEIMER'S DISEASE, SCHIZOPHRENIA, LATERAL AMYOTROPHIC SCLEROSIS OR HUNTINGTON'S CHOREA. LES LABORATORIES SERVIER (FR) 2002-07-16 US disclosed