SCHEMBL7742769

SCHEMBL7742769

O=c1[nH]c2cc(F)c(-c3ccc(C(F)(F)F)cc3)cc2cc1P(=O)(O)O

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.39
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
KIF11 P52732 1/20 0.35
COMT P21964 1/20 0.34
GPR35 Q9HC97 1/20 0.34
TNKS O95271 2/20 0.33
TNKS2 Q9H2K2 2/20 0.33
PARP1 P09874 2/20 0.33
WNT3A P56704 1/20 0.33
TYMS P04818 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6940851 0.87 TNKS (0.39) CDK5CDK5R1COMTTNKS
SCHEMBL7739889 0.82 APP (0.35) APPCDK5CDK5R1AKR1C3AKR1C2
SCHEMBL7739895 0.82 AKR1C3 (0.36) APPCDK5CDK5R1AKR1C3AKR1C2
SCHEMBL8828097 0.77 DAO (0.37)
SCHEMBL7741405 0.77 NTRK1 (0.38)
SCHEMBL7740551 0.76 PRKAG1 (0.43)
SCHEMBL6935464 0.71 PRKAG1 (0.43)
SCHEMBL7740618 0.71 PTGES (0.38) AKR1C3AKR1C2TNKS
SCHEMBL7740617 0.70 PTGES (0.36) CDK5CDK5R1TNKSTYMS
SCHEMBL7742754 0.70 PRKAG1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420386-B1 SPINAL TRAUMATISM, EPILEPSY, CHRONIC NEURODEGENERATIVE DISEASES SUCH AS ALZHEIMER'S DISEASE, SCHIZOPHRENIA, LATERAL AMYOTROPHIC SCLEROSIS OR HUNTINGTON'S CHOREA. LES LABORATORIES SERVIER (FR) 2002-07-16 US disclosed