SCHEMBL7739895

SCHEMBL7739895

CCC(C)OP(=O)(O)c1cc2cc(-c3ccc(C(F)(F)F)cc3)c(F)cc2[nH]c1=O

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.36
AKR1C2 P52895 2/20 0.36
APP P05067 1/20 0.34
GRIN1 Q05586 1/20 0.33
PDE2A O00408 5/20 0.33
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
TYMS P04818 1/20 0.32
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7740618 0.90 PTGES (0.38) AKR1C3AKR1C2GRIN1PDE2A
SCHEMBL6929181 0.84 GRIN1 (0.39) GRIN1PDE2ACDK5CDK5R1
SCHEMBL7735090 0.82 NTRK1 (0.36) AKR1C3AKR1C2PDE2A
SCHEMBL7742769 0.82 APP (0.39) AKR1C3AKR1C2APPCDK5CDK5R1
SCHEMBL7739647 0.81 PRKAG1 (0.38)
SCHEMBL7739889 0.81 APP (0.35) AKR1C3AKR1C2APPPDE2ACDK5
SCHEMBL6928605 0.79 HPRT1 (0.31) GRIN1
SCHEMBL7198441 0.79 AR (0.36) GRIN1
SCHEMBL7741122 0.78 PRKAG1 (0.38) GRIN1
SCHEMBL6923316 0.78 GRIN1 (0.36) GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420386-B1 SPINAL TRAUMATISM, EPILEPSY, CHRONIC NEURODEGENERATIVE DISEASES SUCH AS ALZHEIMER'S DISEASE, SCHIZOPHRENIA, LATERAL AMYOTROPHIC SCLEROSIS OR HUNTINGTON'S CHOREA. LES LABORATORIES SERVIER (FR) 2002-07-16 US disclosed