SCHEMBL7740294

SCHEMBL7740294

COCc1c(C(=O)C#Cc2ccccc2)cnn1-c1ccnc2cc(Cl)ccc12

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.40
NTSR1 P30989 5/20 0.40
IDE P14735 1/20 0.40
NPC1 O15118 1/20 0.39
PTGS1 P23219 1/20 0.39
CYP2C19 P33261 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
CLK1 P49759 1/20 0.39
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
FFAR1 O14842 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744802 0.85 CCR5 (0.47) CCR5NTSR1IDENPC1PTGS1
SCHEMBL7745260 0.80 NTSR1 (0.42) CCR5NTSR1IDEKDM4EMAPT
SCHEMBL7740114 0.79 IDE (0.45) CCR5IDEPTGS1CYP2C19PTGDR2
SCHEMBL7745262 0.79 CCR5 (0.43) CCR5IDENPC1PTGS1CYP2C19
SCHEMBL7740033 0.79 IDE (0.52) CCR5NTSR1IDEPTGS1CYP2C19
SCHEMBL7744853 0.79 MAPT (0.46) CCR5NTSR1IDEKDM4EMAPT
SCHEMBL7744743 0.78 CCR5 (0.43) CCR5NTSR1IDEKDM4EMAPT
SCHEMBL7745238 0.78 CCR5 (0.42) CCR5IDENPC1PTGS1CYP2C19
SCHEMBL7744835 0.78 IDE (0.46) CCR5IDEPTGS1CYP2C19PTGDR2
SCHEMBL7745335 0.78 KMT2A (0.45) CCR5NTSR1IDEKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001002385-A1 1-(QUINOLIN-4-YL)-1H-PYRAZOLE DERIVATIVES AND THEIR USE AS FUNGICIDES AVENTIS CROPSCIENCE S.A. (FR) 2001-01-11 WO claimed
WO-2001002385-A1 1-(QUINOLIN-4-YL)-1H-PYRAZOLE DERIVATIVES AND THEIR USE AS FUNGICIDES AVENTIS CROPSCIENCE S.A. (FR) 2001-01-11 WO disclosed