SCHEMBL7740469

SCHEMBL7740469

CCSC(=N)Nc1ccc(-n2cc(C)cn2)c(CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.34
HDAC10 Q969S8 1/20 0.34
NAMPT P43490 2/20 0.33
RAF1 P04049 1/20 0.33
BRAF P15056 1/20 0.33
SCD O00767 1/20 0.33
RORC P51449 8/20 0.33
HDAC1 Q13547 1/20 0.33
GLS O94925 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
MAPKAPK2 P49137 1/20 0.32
CCKBR P32239 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
MAPK1 P28482 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7740424 0.85 MEN1 (0.36) HDAC6HDAC10NAMPTRORCGLS
SCHEMBL7738859 0.81 HDAC6 (0.36) HDAC6HDAC10NAMPTRAF1BRAF
SCHEMBL7740476 0.80 NOS1 (0.38) HDAC6HDAC10CA12CA1CA2
SCHEMBL27564255 0.80 NTRK1 (0.31) PIK3CAPIK3CG
Hydrochloric Acid SCHEMBL27512818 0.79 TDO2 (0.32) PIK3CAPIK3CG
SCHEMBL27564542 0.78 JAK2 (0.39) NAMPTHDAC1GLS
SCHEMBL27577235 0.78 IDO1 (0.43) HDAC6HDAC10NAMPTHDAC1GLS
SCHEMBL27564508 0.75 ALDH1A1 (0.44) NAMPTGLS
SCHEMBL27544136 0.73 IDO1 (0.41) NAMPTHDAC1GLSCA12CA1
SCHEMBL27564883 0.72 CYP2C9 (0.45) NAMPTHDAC1GLSCYP2C9MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN disclosed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed