SCHEMBL7740717

SCHEMBL7740717

COc1ccc2c(c1)nc(Cl)n2[C@@H]1O[C@H](C)[C@@H](O)[C@H]1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.38
PRKACA P17612 1/20 0.38
RPS6KB1 P23443 1/20 0.38
GSK3B P49841 1/20 0.38
ROCK1 Q13464 1/20 0.38
IDH1 O75874 3/20 0.37
ALDH1A1 P00352 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
SLC5A1 P13866 2/20 0.36
SLC5A2 P31639 2/20 0.36
ADK P55263 1/20 0.36
POLB P06746 1/20 0.36
HTT P42858 1/20 0.36
HTR3A P46098 1/20 0.36
ACSS2 Q9NR19 1/20 0.36
PDE2A O00408 2/20 0.35
PDE10A Q9Y233 2/20 0.35
HSPA8 P11142 1/20 0.35
KDM4E B2RXH2 2/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7734310 0.81 HDAC6 (0.50) TDP1PRKACARPS6KB1GSK3BROCK1
SCHEMBL7740696 0.80 ALDH1A1 (0.36) TDP1PRKACARPS6KB1GSK3BROCK1
SCHEMBL7739180 0.80 HDAC6 (0.49) ADKHSPA8ADORA3
SCHEMBL7739934 0.80 HDAC6 (0.49) ADKHSPA8ADORA3
SCHEMBL7124713 0.80 HDAC6 (0.49) ADKHSPA8ADORA3
SCHEMBL7739177 0.80 HDAC6 (0.49) ADKHSPA8ADORA3
SCHEMBL7739913 0.73 SLC15A1 (0.38) ADKHSPA8KMT2AADORA3
SCHEMBL7734525 0.69 HDAC6 (0.57) ADKHTTHSPA8KMT2A
SCHEMBL25443596 0.69 ALDH1A1 (0.55) TDP1ALDH1A1SMN1; SMN2POLBHTT
SCHEMBL8189109 0.68 HDAC6 (0.51) ADKHSPA8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6413938-B1 HERPES VIRUS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2002-07-02 US disclosed
EP-0970100-A1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 2000-01-12 EP disclosed
WO-1998035977-A1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 1998-08-20 WO disclosed