SCHEMBL7740832

SCHEMBL7740832

C=CC[Si](C)(C)c1cc(CC(NC(=O)NOC(C)(C)C)C(=O)OC)c2ccccc2c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.36
KMT2A Q03164 4/20 0.35
MEN1 O00255 2/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
PSMB8 P28062 2/20 0.34
PSMB5 P28074 2/20 0.34
TACR1 P25103 1/20 0.34
TACR3 P29371 1/20 0.34
HCRTR1 O43613 1/20 0.34
MAPT P10636 1/20 0.33
NLRP3 Q96P20 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7738440 0.86 TACR1 (0.46) KMT2AMEN1ALDH1A1LMNATACR1
SCHEMBL7738442 0.86 TACR1 (0.46) KMT2AMEN1ALDH1A1LMNATACR1
SCHEMBL7739255 0.80 ATM (0.41) ATMKMT2AMEN1ALDH1A1LMNA
SCHEMBL7739221 0.77 ATM (0.33) ATMKMT2AMEN1ALDH1A1LMNA
SCHEMBL7738397 0.75 NR1H2 (0.38) KMT2AL3MBTL1
SCHEMBL20240283 0.70 KMT2A (0.58) ATMKMT2AMEN1ALDH1A1LMNA
SCHEMBL20240285 0.65 CTSS (0.50) ATMKMT2AMEN1ALDH1A1LMNA
SCHEMBL7738441 0.64 AKR1B1 (0.32) ALDH1A1TACR1
SCHEMBL7738409 0.64 NOS2 (0.43) ATMKMT2AALDH1A1TACR1L3MBTL1
SCHEMBL7738402 0.64 NOS2 (0.43) ATMKMT2AALDH1A1TACR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6416861-B1 COMBINATORIAL CHEMISTRY NORTHWESTERN UNIVERSITY 2002-07-09 US disclosed