SCHEMBL7743428

SCHEMBL7743428

COCc1nc(=O)n(C(=O)NCCCN2CCC3(CC2)CN(S(C)(=O)=O)c2cc(F)ccc23)c(-c2ccc(F)c(F)c2)c1C(=O)OC

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 20/20 0.39
ADRA1D P25100 19/20 0.39
ADRA1B P35368 19/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7743413 0.93 ADRA1D (0.42) ADRA1AADRA1DADRA1B
SCHEMBL7749103 0.76 ADRA1D (0.43) ADRA1AADRA1DADRA1B
SCHEMBL7748895 0.71 CCR2 (0.44) ADRA1AADRA1DADRA1B
SCHEMBL7750602 0.66 CCR2 (0.41) ADRA1AADRA1DADRA1B
SCHEMBL8143724 0.63 ADRA1D (0.61) ADRA1AADRA1DADRA1B
SCHEMBL7534012 0.59 ADRA1A (0.86) ADRA1AADRA1DADRA1B
SCHEMBL8138620 0.59 ADRA1D (0.53) ADRA1AADRA1DADRA1B
SCHEMBL31396115 0.59 NPY5R (0.47)
SCHEMBL8135445 0.58 ADRA1D (0.45) ADRA1AADRA1DADRA1B
SCHEMBL6214008 0.58 NPY5R (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001022919-A2 SPIRO[BICYCLIC -AZACYCLOALKYL AND -CYCLOALKYL] DERIVATIVES AND USES THEREOF MERCK & CO., INC. (US) 2001-04-05 WO claimed