SCHEMBL7749103

SCHEMBL7749103

COCc1nc(=O)n(C(=O)NCCCN2CCC3(CC2)OC(=O)Nc2ccc(Cl)cc23)c(-c2ccc(F)c(F)c2)c1C(=O)OC

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 17/20 0.43
ADRA1A P35348 17/20 0.43
ADRA1B P35368 17/20 0.43
CCR2 P41597 3/20 0.42
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7750602 0.90 CCR2 (0.41) ADRA1DADRA1AADRA1BCCR2TDP1
SCHEMBL7748895 0.84 CCR2 (0.44) ADRA1DADRA1AADRA1BCCR2TDP1
SCHEMBL7743413 0.77 ADRA1D (0.42) ADRA1DADRA1AADRA1B
SCHEMBL7743428 0.76 ADRA1A (0.39) ADRA1DADRA1AADRA1B
SCHEMBL7747425 0.73 ADRA1A (0.49) ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL7748897 0.73 ADRA1A (0.51) ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL7748890 0.73 ADRA1A (0.51) ADRA1DADRA1AADRA1B
SCHEMBL7743434 0.66 CCR2 (0.39) ADRA1DADRA1AADRA1BCCR2TDP1
SCHEMBL7743435 0.66 CCR2 (0.39) ADRA1DADRA1AADRA1BCCR2TDP1
SCHEMBL8143724 0.64 ADRA1D (0.61) ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001022919-A2 SPIRO[BICYCLIC -AZACYCLOALKYL AND -CYCLOALKYL] DERIVATIVES AND USES THEREOF MERCK & CO., INC. (US) 2001-04-05 WO disclosed