SCHEMBL7748895

SCHEMBL7748895

COCc1nc(=O)n(CCCCCN2CCC3(CC2)OC(=O)Nc2ccc(F)cc23)c(-c2ccc(F)c(F)c2)c1C(=O)OC

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 3/20 0.44
TDP1 Q9NUW8 1/20 0.38
PLD2 O14939 3/20 0.37
PLD1 Q13393 3/20 0.37
ADRA1D P25100 14/20 0.36
ADRA1A P35348 14/20 0.36
ADRA1B P35368 14/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7750602 0.94 CCR2 (0.41) CCR2TDP1PLD2PLD1ADRA1D
SCHEMBL7749103 0.84 ADRA1D (0.43) CCR2TDP1ADRA1DADRA1AADRA1B
SCHEMBL7743428 0.71 ADRA1A (0.39) ADRA1DADRA1AADRA1B
SCHEMBL4999331 0.69 CCR2 (0.49) CCR2TDP1PLD2PLD1ADRA1A
SCHEMBL4999332 0.69 CCR2 (0.49) CCR2TDP1PLD2PLD1ADRA1A
SCHEMBL7748936 0.68 CCR2 (0.43) CCR2TDP1PLD2PLD1ADRA1D
SCHEMBL7743413 0.67 ADRA1D (0.42) ADRA1DADRA1AADRA1B
SCHEMBL631540 0.66 PLD2 (0.51) CCR2TDP1PLD2PLD1
SCHEMBL631177 0.65 TACR3 (0.49) CCR2PLD2PLD1
SCHEMBL13864851 0.65 CCR2 (0.50) CCR2TDP1PLD2PLD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001022919-A2 SPIRO[BICYCLIC -AZACYCLOALKYL AND -CYCLOALKYL] DERIVATIVES AND USES THEREOF MERCK & CO., INC. (US) 2001-04-05 WO disclosed