SCHEMBL7748837

SCHEMBL7748837

CCc1ccnc(CCN(C)C)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.48
NOS1 P29475 1/20 0.48
NOS2 P35228 1/20 0.48
KDM4E B2RXH2 2/20 0.46
TSHR P16473 2/20 0.46
POLB P06746 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
HTR1A P08908 1/20 0.46
HTR1D P28221 1/20 0.46
HTR1B P28222 1/20 0.46
CHRNA7 P36544 1/20 0.41
TAAR1 Q96RJ0 6/20 0.39
HRH3 Q9Y5N1 3/20 0.39
HTR6 P50406 1/20 0.38
LMNA P02545 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
RECQL P46063 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17828159 0.81 NOS3 (0.52) NOS3NOS1NOS2KDM4ETSHR
SCHEMBL19160064 0.81 TSHR (0.47) NOS3NOS1NOS2KDM4ETSHR
SCHEMBL10066451 0.80 NOS3 (0.55) NOS3NOS1NOS2KDM4ETSHR
SCHEMBL13337725 0.80 NOS3 (0.55) NOS3NOS1NOS2KDM4ETSHR
Hydrochloric Acid SCHEMBL11420925 0.79 NOS3 (0.53) NOS3NOS1NOS2KDM4ETSHR
SCHEMBL21657227 0.78 HRH3 (0.39) KDM4ETSHRPOLBTDP1HTR1A
SCHEMBL31644385 0.78 TAAR1 (0.49) KDM4ECHRNA7TAAR1HRH3LMNA
SCHEMBL218290 0.78 NOS3 (0.61) NOS3NOS1NOS2KDM4ETSHR
SCHEMBL2552826 0.77 NOS2 (0.52) NOS3NOS1NOS2KDM4ETSHR
SCHEMBL5340892 0.77 NOS3 (0.57) NOS3NOS1NOS2KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1069901-A4 CALCILYTIC COMPOUNDS AND METHOD OF USE SMITHKLINE BEECHAM CORP (US) 2001-06-13 EP disclosed
EP-1069901-A1 CALCILYTIC COMPOUNDS AND METHOD OF USE SMITHKLINE BEECHAM CORPORATION (US) 2001-01-24 EP disclosed
WO-1999051241-A1 CALCILYTIC COMPOUNDS AND METHOD OF USE SMITHKLINE BEECHAM CORPORATION (US) 1999-10-14 WO disclosed