SCHEMBL7750256

SCHEMBL7750256

COc1cc(OC(N)=O)c(Cl)cc1-c1nn(C2CCNC2)c(=O)o1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SUV39H2 Q9H5I1 5/20 0.35
PIK3CD O00329 1/20 0.35
ABL1 P00519 1/20 0.35
EGFR P00533 1/20 0.35
HCK P08631 1/20 0.35
SRC P12931 1/20 0.35
KDR P35968 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
MTOR P42345 1/20 0.35
PIK3CG P48736 1/20 0.35
EPHB4 P54760 1/20 0.35
PRKDC P78527 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
HTR2C P28335 3/20 0.34
HTR2B P41595 3/20 0.34
HTR2A P28223 1/20 0.34
S1PR2 O95136 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6958303 0.83 DRD4 (0.41) SUV39H2PIK3CDABL1EGFRHCK
SCHEMBL8304880 0.80 HTR4 (0.44) SUV39H2HTR4HTR3A
Bromide SCHEMBL8366387 0.79 HTR4 (0.43) SUV39H2HTR4HTR3A
SCHEMBL8368075 0.78 MAPT (0.40) SUV39H2HPGD
SCHEMBL8308838 0.77 DRD4 (0.38) SUV39H2HPGDHTR4
SCHEMBL7808395 0.71 HTR4 (0.45) HTR4
SCHEMBL8368080 0.70 FAAH (0.43) SRCKDR
SCHEMBL8305104 0.70 HTR4 (0.44) HTR4
Bromide SCHEMBL7937589 0.70 HTR4 (0.45) HTR4
SCHEMBL8366414 0.70 MAPT (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248757-B1 ANTISEROTONINE AGENTS SANOFI-SYNTHELABO (FR) 2001-06-19 US disclosed
EP-0980368-A1 3-(PYRROLIDIN-3-YL)-1,3,4-OXADIAZOL-2(3H)-ONE DERIVATIVES AND THEIR USE AS 5-HT4 LIGANDS SANOFI-SYNTHELABO (FR) 2000-02-23 EP disclosed
WO-1998050381-A1 3-(PYRROLIDIN-3-YL)-1,3,4-OXADIAZOL-2(3H)-ONE DERIVATIVES AND THEIR USE AS 5-HT4 LIGANDS SANOFI-SYNTHELABO (FR) 1998-11-12 WO disclosed