SCHEMBL6958303

SCHEMBL6958303

COc1cc(NC(=O)O)c(Cl)cc1-c1nn(C2CCNC2)c(=O)o1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.41
PAICS P22234 2/20 0.35
S1PR2 O95136 1/20 0.35
SUV39H2 Q9H5I1 1/20 0.33
STAT3 P40763 2/20 0.33
ALDH1A1 P00352 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
HPGD P15428 1/20 0.33
MELK Q14680 1/20 0.33
PDE7A Q13946 1/20 0.33
GPR55 Q9Y2T6 2/20 0.33
PIK3CD O00329 1/20 0.33
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33
HCK P08631 1/20 0.33
SRC P12931 1/20 0.33
KDR P35968 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
MTOR P42345 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8308838 0.95 DRD4 (0.38) DRD4PAICSSUV39H2STAT3ALDH1A1
SCHEMBL7799616 0.86 HTR4 (0.36) DRD4STAT3ALDH1A1TDP1HPGD
SCHEMBL8307501 0.85 GPR55 (0.39) DRD4GPR55CNR1
SCHEMBL7799610 0.85 HTR4 (0.38) STAT3ALDH1A1HPGDGPR55
Hydrochloric Acid SCHEMBL7943941 0.84 HTR4 (0.37) TDP1GPR55
SCHEMBL7750256 0.83 SUV39H2 (0.35) S1PR2SUV39H2HPGDMELKPIK3CD
SCHEMBL8305942 0.82 TP53 (0.40) SUV39H2ALDH1A1GPR55CNR1
SCHEMBL8368080 0.81 FAAH (0.43) DRD4ALDH1A1SRCKDRCNR1
SCHEMBL6967209 0.79 DRD4 (0.37) DRD4ALDH1A1TSHR
SCHEMBL8310238 0.79 DRD4 (0.48) DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0980368-B1 3-(PYRROLIDIN-3-YL)-1,3,4-OXADIAZOL-2(3H)-ONE DERIVATIVES AND THEIR USE AS 5-HT4 LIGANDS SANOFI SYNTHELABO (FR) 2003-10-22 EP disclosed
US-6248757-B1 ANTISEROTONINE AGENTS SANOFI-SYNTHELABO (FR) 2001-06-19 US disclosed