SCHEMBL8308838

SCHEMBL8308838

COc1cc(NC(=O)O)c(Cl)cc1-c1nn(C2CCNCC2)c(=O)o1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.38
PAICS P22234 3/20 0.37
ALDH1A1 P00352 2/20 0.35
GPR55 Q9Y2T6 4/20 0.35
CNR1 P21554 2/20 0.35
IRAK4 Q9NWZ3 1/20 0.34
HTR4 Q13639 2/20 0.34
STAT3 P40763 2/20 0.34
HPGD P15428 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
SUV39H2 Q9H5I1 2/20 0.34
NSD3 Q9BZ95 1/20 0.33
TSHR P16473 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6958303 0.95 DRD4 (0.41) DRD4PAICSALDH1A1GPR55CNR1
SCHEMBL8307501 0.89 GPR55 (0.39) DRD4GPR55CNR1IRAK4CNR2
SCHEMBL7799616 0.87 HTR4 (0.36) DRD4ALDH1A1GPR55CNR1HTR4
SCHEMBL7799610 0.86 HTR4 (0.38) ALDH1A1GPR55HTR4STAT3HPGD
SCHEMBL8368080 0.86 FAAH (0.43) DRD4ALDH1A1CNR1
Hydrochloric Acid SCHEMBL7943941 0.85 HTR4 (0.37) GPR55HTR4TDP1
SCHEMBL8305942 0.85 TP53 (0.40) ALDH1A1GPR55CNR1SUV39H2CNR2
SCHEMBL8304880 0.82 HTR4 (0.44) HTR4SUV39H2
Bromide SCHEMBL8366387 0.82 HTR4 (0.43) HTR4SUV39H2
SCHEMBL8310238 0.82 DRD4 (0.48) DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863897-B1 5-PHENYL-3-(PIPERIDIN-4-YL)-1,3,4-OXADIAZOL-2(3H)-ONE DERIVATIVES FOR USE AS 5-HT4- OR H3-RECEPTOR LIGANDS SYNTHELABO (FR) 1999-06-16 EP disclosed