SCHEMBL7756403

SCHEMBL7756403

CC(C)N/C(=N/c1cccc(C(F)(F)F)c1)NC#N

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.48
HTR3B O95264 1/20 0.48
HTR3A P46098 1/20 0.48
HTR3D Q70Z44 1/20 0.48
HTR3C Q8WXA8 1/20 0.48
MAPT P10636 1/20 0.47
NPSR1 Q6W5P4 1/20 0.46
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
NOS3 P29474 2/20 0.43
NOS1 P29475 2/20 0.43
NOS2 P35228 2/20 0.43
ESR1 P03372 2/20 0.43
ESR2 Q92731 2/20 0.43
CTSL P07711 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
KIF11 P52732 1/20 0.41
GAA P10253 1/20 0.39
IDO1 P14902 1/20 0.39
CRHR1 P34998 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7756407 1.00 HTR3E (0.48) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8140971 0.89 ALDH1A1 (0.47) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8143183 0.87 KIF11 (0.42) MAPTNPSR1CYP1A2CYP2C19CTSL
SCHEMBL7756397 0.79 LMNA (0.47) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8134156 0.77 KIF11 (0.41) MAPTNPSR1CYP1A2CYP2C19CTSL
SCHEMBL8136535 0.75 KIF11 (0.39) MAPTNPSR1CYP1A2CYP2C19CTSL
SCHEMBL9298624 0.73 KIF11 (0.54) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL11165566 0.72 HTR3E (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7756412 0.72 ABCC9 (0.55) MAPTNPSR1CYP1A2CYP2C19SMN1; SMN2
SCHEMBL7753800 0.71 KMT2A (0.57) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077933-A1 SUBSTITUTED GUANIDINES AND DIAMINONITROETHENES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 2001-02-28 EP disclosed
US-6147098-A USEFUL IN THE TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM, CARDIOVASCULAR SYSTEM, PULMONARY SYSTEM, GASTROINTESTINAL SYSTEM AND ENDOCRINOLOGIC SYSTEM NOVO NORDISK A/S (DK) 2000-11-14 US disclosed
WO-1999058497-A1 SUBSTITUTED GUANIDINES AND DIAMINONITROETHENES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1999-11-18 WO disclosed